GAZI UNIVERSITY INFORMATION PACKAGE - 2019 ACADEMIC YEAR

COURSE DESCRIPTION
PRODRUGS AND PRODRUG DESIGN/FKİ-3180
Course Title: PRODRUGS AND PRODRUG DESIGN
Credits 2 ECTS 5
Course Semester 1 Type of The Course Elective
COURSE INFORMATION
 -- (CATALOG CONTENT)
 -- (TEXTBOOK)
 -- (SUPPLEMENTARY TEXTBOOK)
 -- (PREREQUISITES AND CO-REQUISITES)
 -- LANGUAGE OF INSTRUCTION
  Turkish
 -- COURSE OBJECTIVES
 -- COURSE LEARNING OUTCOMES
Have gained knowledge about Prodrugs.

 -- MODE OF DELIVERY
   The mode of delivery of this course is face to face.
 --WEEKLY SCHEDULE
1. Week  Concept of prodrug
2. Week  Classification of prodrug
3. Week  Principles of prodrug desing
4. Week  Bipartat Prodrugs, Tripartat Prodrugs
5. Week  Mutual Prodrugs
6. Week  Fuctional groups of prodrugs
7. Week  Mechanism of prodrugs
8. Week  Roles of hydrolytic enzymes in prodrugs
9. Week  Midterm exam
10. Week  Macromolecular drug carrier systems
11. Week  Bioprecursor prodrugs
12. Week  Prodrug development
13. Week  Design of prodrug
14. Week  Use of prodrugs
15. Week  Prodrug strategy
16. Week  Final exam
 -- TEACHING and LEARNING METHODS
 -- ASSESSMENT CRITERIA
 
Quantity
Total Weighting (%)
 Midterm Exams
1
60
 Assignment
1
40
 Application
0
0
 Projects
0
0
 Practice
0
0
 Quiz
0
0
 Percent of In-term Studies  
50
 Percentage of Final Exam to Total Score  
50
 -- WORKLOAD
 Activity  Total Number of Weeks  Duration (weekly hour)  Total Period Work Load
 Weekly Theoretical Course Hours
14
2
28
 Weekly Tutorial Hours
0
 Reading Tasks
6
5
30
 Searching in Internet and Library
5
5
25
 Material Design and Implementation
0
 Report Preparing
0
 Preparing a Presentation
2
2
4
 Presentation
2
5
10
 Midterm Exam and Preperation for Midterm Exam
2
5
10
 Final Exam and Preperation for Final Exam
2
10
20
 Other (should be emphasized)
0
 TOTAL WORKLOAD: 
127
 TOTAL WORKLOAD / 25: 
5.08
 Course Credit (ECTS): 
5
 -- COURSE'S CONTRIBUTION TO PROGRAM
NO
PROGRAM LEARNING OUTCOMES
1
2
3
4
5
1X
2X
3X
4X
5X
6X
7X
8X
9
10X
11X
12
13
14X
15X
16X
 -- NAME OF LECTURER(S)
   (Prof. Dr. Tijen ONKOL)
 -- WEB SITE(S) OF LECTURER(S)
   ( www.gazi.edu.tr/~tijen , )
 -- EMAIL(S) OF LECTURER(S)
   (tijen@gazi.edu.tr , bcalıskan@gazi.edu.tr)